(828) 505-2885 Appointment

Peptide Therapy Serving Greenville, SC

Lead a Thriving Life

“George and his staff are great to work with and very knowledgeable. I’ve had fun learning and doing the peptide program. It’s been very smooth.” - Henry M., Google Review

Peptide Therapy at Biltmore Restorative Medicine and Aesthetics

Peptides play an integral role in bodily processes ranging from cellular functioning to energy burning, weight loss, muscle growth, wound healing, skin health, and mental acuity. With Peptide Therapy Greenville patients can renew their vitality and overall well-being with our A4M peptide-certified practitioners at Biltmore Restorative Medicine and Aesthetics in Asheville.

Asheville peptide therapy model with brown hair

What is Peptide Therapy?


Peptides, tiny chains of amino acids, are present in all living cells. The body makes use of more than 7,000 peptides, each with specific applications that impact biological processes. Administering Peptides in a therapeutic setting can restore balance to the body, allowing it to function as it should so you can thrive.

Peptide Delivery Methods


Our partnerships with cutting-edge pharmacies certified in peptide protocols allow us to compound peptides into injectables, capsules, and creams. Working side-by-side with our specialists, you’ll be able to select the Peptide Therapy that works for you.

Benefits of Peptide Therapy


The human body performs optimally when neurochemicals are balanced harmoniously. If you are feeling off-kilter, that is your first clue that something needs to change. Peptide therapy is a powerful tool you can use to look and feel more like you did when you were young, healthy, energized, and full of life.

Potential Advantages of Peptide Therapy

Here are a few benefits that our Greenville Peptide Therapy patients should take into account:

  • Fat Loss
  • Restful Sleep
  • Stronger Muscles
  • Healthier Hair and Skin
  • Strengthened Immunity
  • Enhanced Sexual Wellness
  • Improved Focus and Memory
  • Faster Tissue Repair and Muscle Recovery

Who is an ideal candidate for Peptide Therapy?

Peptide therapy is safe and effective for many individuals, but there may be instances when it is not appropriate. Your provider at Biltmore Restorative will review your medical history to ensure you are a suitable candidate. During your consultation, you will undergo a detailed assessment to determine if this therapy can benefit you.


Our bespoke Greenville Peptides at Biltmore Restorative can contribute to a better quality of life.


Unbeknownst to them, many people struggling to lose weight have elevated NNMT levels. Scientists have found a powerful NNMT inhibitor called 5-Amino-1MQ can reduce fat deposits that resist conventional diet efforts while lowering cholesterol.


AOD 9404 mimics a growth hormone that regulates fat metabolism. Studies show it stimulates lipolysis, the process of breaking down fat, and inhibits lipogenesis without adversely affecting blood sugar.


The peptide BPC-157 is made of 15 amino acids derived from human gastric acid. BPC, which stands for body protection compound, has a healing effect on wounds, sunburns, tendons, and ligaments. It is also believed to prevent stomach ulcers and increase blood flow to repair damaged tissues. BPC-157 may also stimulate collagen synthesis, decrease inflammation, and improve heart health.


A combination of two peptides, CJC1295/Ipamorelin, consists of a growth hormone-releasing hormone (GHRH) and a growth hormone-releasing peptide (GHRP). Together, they trigger the release of growth hormone while promoting protein synthesis, making it a favorite of athletes seeking to increase muscle mass and burn fat the natural way. Additionally, CJC/Ipamorelin shows positive effects in individuals with poor sleep habits and cognition.


Neurodegenerative diseases like Alzheimer’s, Parkinson’s, and Huntington’s ultimately cause issues with memory recall and motor skills. To potentially improve cognition, we rely on Dihexa, a tiny molecule linked to improved focus and memory.


With age, telomeres tend to shrink leading to cellular and tissue deterioration. Epitalon, an anti-aging peptide, is believed to increase the length of telomeres, potentially slowing the progression of age-related diseases.


GHK-Cu levels drop as we age, slowing wound healing and tissue regeneration. To combat these effects, supplementing with GHK-Cu may improve the health of the skin, hair follicles, bone tissue, and intestinal and stomach linings. It also serves as an antioxidant and anti-inflammatory, increases collagen production, can help promote hair growth, improve hair density, and reduce shedding.


A powerful antioxidant, glutathione, keeps cells healthy by disposing of toxins. Glutathione injections offer a host of benefits, such as reducing oxidative stress, dialing up skin radiance, calming psoriasis symptoms, improving insulin resistance, and more.


LGD-4033 (VK5211) is a non-steroidal selective androgen receptor modulator. This tissue-selective anabolic agent aids in muscle and bony growth and potentially counteracts muscle wasting and cachexia. Since it is not a steroid, it will not adversely affect testosterone or estrogen levels.

Melanotan-II (MT2)

Looking for a darker tan? Consider Melanotan-II, a peptide that increases melanocytes, boosting melanin production naturally. Additionally, it shows potential for reducing body fat and increasing libido.


This novel peptide activates GHSR in the brain, which can have positive effects on mood, sleep, appetite control, cognition, memory, bone density, muscle mass, and growth hormone secretions. It also increases insulin-like growth factor 1 (IGF-1).


MOTS-C is a peptide consisting of 14 amino acids. Classified as a short open reading frame (sORF), it aids in metabolic processes that affect muscle, fat, and insulin sensitivity in individuals living with obesity or diabetes.


NAD+ helps regulate stress levels and plays a role in more than 500 enzymatic reactions that affect biological functioning. Peptides that boost NAD+ may improve vision, hearing loss, motor skills, and cognitive abilities. It may also alleviate symptoms from autoimmune diseases and combat age-related illnesses. Studies show NAD+ boosters can improve liver function, kidney function, skeletal muscles, and blood vessels, as well as repair damaged DNA.


Oxytocin, the “love hormone,” is a neurotransmitter linked to sexual arousal and connection. Research suggests increasing oxytocin may promote better interpersonal relations, lower stress, reduce blood pressure, and increase satisfaction in the bedroom for both men and women.

PT-141 (Bremelanotide)

With age, many people experience a drop in sexual desire, causing disinterest in sex and potentially straining intimate relationships. Taking bremelanotide stimulates a hormone known as melanocortin to enhance sexual arousal and intensify orgasms.


Selank is a synthetic peptide with anxiolytic properties. Clinical data shows it may curb anxiety, fear, stress, and aggression. As a nootropic compound, it also aids in memory and learning. Unlike benzodiazepines, there is no risk of withdrawal or dependence.


Semax has potent neuroprotective, neurorestorative, and nootropic properties. Designed to mimic adrenocorticotropic hormone (ACTH), Semax is found in drugs that treat central nervous system diseases, including ischemic stroke, hypoxia, encephalopathy, glaucoma, and more. Semax may also ease ADHD symptoms, protect the brain against stress, and improve short-term memory.


Mitochondrial dysfunction can lead to disease and cell death. SS-31 may improve mitochondrial health by neutralizing inflammation and free radicals. Able to cross the blood-brain barrier, it is a promising treatment for cognitive and neurodegenerative disorders such as Alzheimer’s, amyotrophic lateral sclerosis (ALS), and Friedreich ataxia.


Those living with neurodegenerative conditions or brain fog may benefit from synapsin. Two ingredients, RG3 and nicotinamide ribose, may improve synaptic plasticity and resistance to neuronal stress, thereby improving memory, decreasing inflammation, and supporting neurological health.


TB-500 is a synthetic version of a peptide called thymosin beta-4, known for its powerful healing potential. It is thought to help repair soft tissue injuries involving the tendons, ligaments, skin, muscles, eyes, and heart.


Tesofensine (NS2330) suppresses appetite and feelings of hunger. It also shows positive effects on fat oxidation, resting energy expenditure, lipoproteins, and triglycerides, making it an excellent option for those struggling to stick to a healthy diet. Tesofensine also helps balance insulin levels and may potentially reverse early type 2 diabetes.


Thymulin is an immune-system-regulating hormone that helps differentiate T lymphocytes and optimize T-helper cells. It also boasts anti-inflammatory properties by reducing cytokines and chemokines while encouraging anti-inflammatory factors such as interleukin-10 (IL-10).


Tirzepatide is studied for its role in treating obesity. Researchers theorize that tirzepatide reduces A1C, making it important for weight loss and cardio-metabolic health. It may also alleviate cravings and, when compounded with Vitamin B12, boost energy levels.

Our Peptide Programs


Our peptides therapy programs at Biltmore Restorative Medicine are fully customizable based on your specific needs and goals.

Weight Management and Fat Loss

Optimizing peptide levels through Peptide Therapy can support your efforts to reach and maintain a healthy weight. When the payoff from counting calories and working out is happening slower than you would like, peptides can accelerate your body’s ability to burn through fat stores, revealing a more toned, streamlined figure over time.

Key Peptides: 5-Amino-1MQ, Tesofensine, AOD-9604, Tirzepatide, CJC/Ipamorelin

Digestive Health, Healing, and Cellular Repair

Chronic injuries and muscle soreness can hold you back from doing the things you love. With Peptide Therapy Greenville patients can accelerate wound healing, relieve muscle pain, instigate cellular repair, heal damaged ligaments, and increase blood circulation. Additionally, peptides for gut health can help resolve issues from a leaky gut, irritable bowel syndrome, Crohn’s disease, and stomach ulcers.

Key Peptides: BPC-157, TB-500, CJC/Ipamorelin, GHK-Cu

Memory and Cognition

Peptides can stimulate nerve regeneration and enhance neuromuscular performance. Patients can sharpen mental acuity, improve concentration, and bolster memory. Medical literature suggests that they may have a beneficial role in managing conditions such as general anxiety, ADHD, opiate withdrawal, Alzheimer’s, Parkinson’s, and ALS.

Key Peptides: NAD+, Dihexa, Epitalon, Semax, Selank, SS-31


Growth hormones steadily decline with age, starting in your 20s. The body’s ability to regenerate and repair tissues takes a hit as a result, leading to weight gain, rapidly aging skin, and hair shedding. Peptides have anti-aging potential, allowing clients to eliminate stubborn fat, improve skin health, and regain fuller hair.

Key Peptides: NAD+, CJC/Ipamorelin, Epitalon, GHK-Cu

Sleep Quality

A restful night of sleep sets the foundation for a great day. If you have difficulty falling asleep or wake up feeling tired, peptides may be the key to a more restorative sleep.

Key Peptides: CJC/Ipamorelin, Epitalon

Skin and Hair Health

Collagen and elastin loss over the years, combined with sun exposure and lifestyle habits like smoking, can exacerbate skin aging, making you look older and more tired than you would like. Peptides may support the skin’s ability to produce collagen, improve fine lines, brighten dull skin, and soften the appearance of scars. For healthy hair, peptide GHK-Cu aids scalp health, promoting thicker hair with less breakage.

Key Peptides: GHK-Cu, Thymulin, Melanotan-2, TB-500

Libido and Sexual Wellness

Peptides can balance neurochemicals within the body and increase dopamine secretion, enhancing sexual desire and relieving uncomfortable symptoms caused by hormonal imbalances in men and women alike. The “neuro-aphrodisiac” effects from peptide injections are proven to amplify intracellular signaling, intensifying sexual satisfaction. Key Peptides: PT-141, Oxytocin

Key Peptides: PT-141, Oxytocin


Peptides are integral to a strong immune system. For example, thymulin is a biocompatible man-made hormone that may improve T-cell function to ward off disease. Early research shows NAD+ can minimize inflammation and may help fight off COVID-19. Those with diabetes, cardiovascular problems, and infections naturally have lower levels of this peptide; Replacing it can promote a higher quality of life.

Key Peptides: Thymulin, NAD+

Muscle Recovery and Performance Enhancement

You work hard in the gym to stay fit. Reward yourself and maximize your workout efforts with peptides proven to increase stamina and aid in muscle recovery. By awakening natural growth hormones within the body, our peptides make it easier to build lean muscle, reduce body fat, turbocharge energy levels, and relieve soreness after workouts.

Key Peptides: MK-677, CJC/Ipamorelin, NAD+

Schedule Your Greenville, SC Peptide Therapy Consultation at Biltmore Restorative Sexual Wellness and Aesthetics Today


At Biltmore Restorative Medicine and Aesthetics, our holistic approach to wellness allows us to help patients radically transform their lives while looking and feeling healthier. Take advantage of our expertise and innovative therapies to get started on building the life you want. For our patients in Greenville Peptide Therapy in a state-of-the-art office is just a short commute away.

Schedule Your Consultation

Biltmore Restorative Medicine and Aesthetics was built for you. We know you don’t trust your look to just anyone. You want the best. Our experienced and industry-leading regenerative medicine providers give you unparalleled personal care and will help you maximize your vitality for years to come.

By submitting this you agree to be contacted by Biltmore Restorative Medicine via text, call or email. Standard rates may apply. For more details, read our Privacy Policy.